Publications in 2011

  1. Ivachtchenko A.V., Yamanushkin P.M., Mitkin O.D., Leneva I.A., Fedyakina I.T. Synthesis and biological activity functionally substituted indole-3-acetic acid. Chem. Pharm. J., 2011, 45 (5), 3-8.

  2. Ivachtchenko A.V., Golovina E.S., Kadieva M.G., Kysil V.M., Mitkin O.D., Tkachenko S.E., Okun I.M. Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists. Bioorg. Med. Chem. 2011, 19, 1482–1491.

  3. Ivachtchenko A.V., Golovina E.S., Kadieva M.G., Koryakova A.G., Mitkin O.D., Tkachenko S.E., Kysil V.M., Okun I.M. 2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: New series of highly potent and specific serotonin 5-HT6 receptor antagonists. Eur. J. Med. Chem., 2011, 46, 1189-1197.

  4. Ivachtchenko A.V., Golovina E.S., Kadieva M.G., Kysil V.M., Mitkin, O.D., Tkachenko S.E., Okun I.M. Synthesis and Structure Activity Relationship (SAR) of (5,7-disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6 Receptor (5-HT6R) Antagonists. J. Med. Chem., 2011, 54, 8161-8173.