Publications in 2012

  1. Pavlov A.V., Veretennikov E.A., Laskin B.M., Ivanenkov Y.A. Potential innovative antibiotics – (R`-benzyl) – (R-tetrazol-1-yl-phenyl) -amine. II-d International Conference “Models of innovative development of the pharmaceutical and medical industry on the basis of universities, as an integrator of science and industry”, MPTI, Dolgoprudny, 15-16 May 2012.

  2. Ivachtchenko A.V., Ivanenkov Y.A. 5HT6 receptor modulators: a patent update. Part 1. Sulfonyl derivatives (Review). Expert Opin. Ther. Pat., 2012, 22(8), 917-964.

  3. Ivachtchenko A.V., Ivanenkov Y.A., Skorenko A.V. 5-HT6 receptor modulators: a patent update. Part 2. Diversity in heterocyclic scaffolds (Review). Expert Opin. Ther. Pat., 2012, 22(10), 1123-1168.

  4. Ivachtchenko A.V., Golovina E. S, Kadieva M. G., Kysil V. M., Mitkin O. D., Vorobiov A.A., Okun I.M. Antagonists of 5-HT6 receptors. Substituted 3-(phenylsulfonyl)-pyrazolo[1,5-a]pyrido[3,4-e]pyrimidines and 3-(phenylsulfonyl)-pyrazolo[1,5-a]pyrido[4,3-d]pyrimidines — synthesis and «structure – activity» relationship. Bioorg. Med. Chem. Lett., 2012, 22, 4273-4280.

  5. Ivachtchenko A.V., Golovina E. S, Kadieva M. G., Mitkin O. D., Tkachenko S.E., Okun I.M. Antagonists of the 5-HT6 receptor. I. Screening of samples of structurally diverse heterocyclic compounds containing a sulfonyl moiety. Chem. Pharm. J., 2012, 46 (5), 48-58.

  6. Ivachtchenko A.V., Golovina E. S, Kadieva M. G., Mitkin O. D., Okun I.M. Antagonists of serotonin receptor subtype 5-HT6. II. The relationship structure – activity (4-phenylsulfonyl-oxazol-5-yl) amine. Chem. Pharm. J., 2012, 46 (11), 55-62.

  7. Ivachtchenko A.V., Golovina E. S, Kadieva M. G., Kysil V. M., Mitkin O. D. Antagonists of serotonin receptor subtype 5-HT6. III. Synthesis and interconnection structure – activity amines containing 3- (arylsulfonyl) -2- (methylthio) pyrazolo [1,5-a] pyrimidine moiety. Chem. Pharm. J., 2012, 46 (10), 40-47.

  8. Ivachtchenko A.V., Golovina E. S, Kadieva M. G., Kysil V. M., Mitkin O. D., Okun I.M. Antagonists of serotonin receptor subtype 5-HT6. IV. Synthesis and relationship of the structure – activity of 3-aryl sulfonyl-2-methyl sulfonyl-pyrazol [1,5-a] pyrimidine, containing the 6-position substituent comprising an amino group. Chem. Pharm. J., 2012, 46 (6), 36-45.

  9. Ivachtchenko A.V., Golovina E. S, Kadieva M. G., Kysil V. M., Mitkin O. D., Okun I.M. Antagonists of serotonin receptor subtype 5-HT6. V. Synthesis, the relationship structure – Activity pyridine substituted 3- (phenylsulfonyl) pyrazolo [1,5-a] pyrimidine. Chem. Pharm. J., 2012, 46 (7), 55-59.