Cancer
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4400 compounds
Covalent serine binders library, 10 warhead scaffolds 4 400 compounds
30000 compounds
Proteolytic enzymes are crucial for a variety of biological processes in organisms ranging from lower to higher organisms. Proteases cleave proteins into smaller fragments by catalyzing peptide bonds hydrolysis.
1400 compounds
The library contains 1400 compounds that seems to be analogues of approved drugs.
5,886 compounds
SH2 PTB domains Focused Library is a set of inhibitors. SH2 and PTB are small protein modules that mediate PPIs involved in signal transduction pathways.
31,972 compounds
Serine Proteases Inhibitors Library is a set of small-molecule compounds that target serine proteases and can be used in anticancer drug discovery.
1,156 compounds
Purine Based Nucleoside Mimetics Library is nucleoside analogues that mimic metabolic purines. They are extracellular messengers and endogenous modulators.
36,324 compounds
Protein Kinases Inhibitors Library is modulators that are used in cancer and inflammation treatment.
31,000 compounds
PRMT Library is set of small-molecule compounds with reported affinity against cancer-assosiated PRMTs.
2,081 compounds
Proline Kinase Library is a set of kinase inhibitors. These kinases play a crucial role in diverse cellular processes and human diseases.
19,000 compounds
PI3K-Targeted Library is a set of small-molecule inhibitors of PI3K signaling pathway. They can be used in effective inhibiting tumor progression.
491 compounds
PD-1/L1 Library is a set of PD-1 and PD-L1 inhibitors. It is a group of anticancer drugs that block the activity of immune checkpoint proteins.
2,292 compounds
Nucleoside Mimetics Library is a set of modified nucleosides that are used as antiviral and antitumor drugs. They were also designed for HIV therapy.
9,000 compounds
Nucleic Acid Ligands is a set of minor and major groove DNA or RNA binders. Such small molecules have proven to be effective antiviral and cancer agents.
4,003 compounds
Small molecules that can inhibit NOTUM thus potentially treating diseases caused by dysregulation of Wnt signaling.
4,805 compounds
MEF2-HDAC (class II) Modulators Library is a set of drug-like compounds aimed at modulating PPI of MEF2 with HDAC involved in physiological processes.
23,319 compounds
MDM2-p53 Interaction Inhibitors Library is a set of drug-like compounds aimed at modulating PPI of MDM2 with p53 involved in tumorigenesis.
9298 compounds
Lysine-specific histone demethylases (KDM) Library
16,000 compounds
KRAS-Targeted Library is a set of novel KRAS-active compounds.
8,000 compounds
Inhibitors of beta-Catenin Signaling is small molecules that target PPI of beta-catenin with other proteins involved in significant physiological processes.
10,991 compounds
Heat shock protein 90 Targeted Library is a set of small-molecule modulators that inhibit the activity of HSP90/70 and can be used as anticancer drugs.
2,230 compounds
Developmental Pathway Hh/Wnt Set is inhibitors of the Hedgehog and Wnt-signaling pathways implicated in cancer.
7,801 compounds
Set of small-molecule compounds that can target cysteine proteases and be used in drug development for cancer, viral, infections treatment.
5,000 compounds
Carbonic anhydrase II library is a set of compounds belonging to the sulfonamides, mercaptans and phenols aimed at modulating of Carbonic anhydrase II activity
15,080 compounds
Molecules from c-Met Library target receptor tyrosine kinase. It prevents binding hepatocyte growth factor with c-Met which can lead to cancer.
11,568 compounds
Bcl2 PPI Inhibitors Library is small molecules that inhibit regulators of programmed cell death.
4,550 compounds
Autophagy-Targeted Library is a set of small-molecule modulators for the regulation of autophagy.
10,000 compounds
Set of small-molecule serine/threonine kinases family inhibitors.
18,000 compounds
Antimitotic Tubulin Library is a set of small-molecule tubulin binders. These inhibitors are potential antimitotic drugs for anticancer therapy.
65,000 compounds
Anticancer Library is a set of small-molecule compounds with anticancer activity and vast target space.
17,000 compounds
Angiogenesis Library is a set of small-molecule compounds that target proteins involved in new blood vessels forming.
4,244 compounds
Androgen Receptor Antagonists Library is a set of non-steroidal small molecules for prostate cancer treatment.
26,000 compounds
Small‐molecule allosteric kinase modulators that target allosteric pockets of kinases outside the conserved ATP‐binding pocket.
15,000 compounds
Akt Targeted Library is a set of small-molecule inhibitors of the Akt-signaling network. These inhibitors are widely used in cancer treatment.
20,000 compounds
microRNAs (miRs) are small (~18e25 nucleotides)
12,206 compounds
Set of small-molecule compounds that inhibit MCL1 thus restoring the apoptotic pathway in tumor cells.
21000 compounds
Adenosine Receptors Targeted Library is a set of small-molecule ligands. They can be used for treating neurodegeneration diseases.
12,000 compounds
Diacylglycerol kinase Inhibitors Library is a set of small-molecules that can inhibit the progression of cancer and innate cytotoxic immunocytes.
8,600 compounds
Chelators targeting matrix metalloproteinases are small-molecule that inhibit proteolytic activity of tumor cells and prevent metastasis.
3,900 compounds
RPTP Targeted Library is small-molecule inhibitors. Disruption of protein tyrosine phosphorylation contributes to a variety of human diseases.
32,596 compounds
PTPN Targeted Library is a set of small-molecule inhibitors. Protein tyrosine phosphatases are important signaling molecules in cell proliferation.
6,767 compounds
Set of RAR receptor antagonists. The retinoic acid receptor is a type of nuclear receptor which can also act as a transcription factor.
5,000 compounds
Glucocorticoid Receptors Library is small-molecule selective modulators of GR which regulates gene transcription.
5,939 compounds
STING Agonist Library is small-molecules that bind and activate STING and lead to IFN production. Can be used in cancer immunotherapy.
1,708 compounds
Integrin Receptors Targeted library is a set of RGD peptides or peptidomimetics that affect many events in tumor cells thereby directly induce apoptosis.
6,000 compounds
Indoleamine 2,3-dioxygenase1 Focused Library is a set of small-molecule compounds that can inhibit inappropriate IDO activity in tumours.
5,000 compounds
BRD4 Targeted Library is a set of small-molecule compounds that inhibit transcriptional and epigenetic regulator - BRD4.
2,016 compounds
Arginase Targeted Library is a set of small-molecule compounds against arginase. This enzyme is implicated in cancer immunosuppression and tumor growth.
20,563 compounds
Spiro Library is a set of scaffolds with twisted structure of two or more rings for the design of new therapeutic agents.
12,000 compounds
SH2 Domain Library is a set of inhibitors. SH2 are modular units, which bind to tyrosyl-phosphorylated peptide on their target protein mediating PPI.
214,102 compounds
PPI Library is a set of small-molecule modulators that have been designed for disrupting PPI and reducing its drawbacks.
23,722 compounds
PPI Tripeptide Mimetics Library is small-molecule PPI inhibitors that mimic significant endogenous tripeptides.
2,335 compounds
Macrocycles Library is a set of macrocyclic peptidomimetics that are potential PPI modulators. It is unique spiro and fused scaffolds.
12,103 compounds
Eccentric PPI Library is a set of unusual ring systems (scaffolds) that lie outside the field of (hetero)aromatic systems.
9,487 compounds
Set of PPI modulators. Cyclic lactam amides result from the Ugi reaction of bifunctional keto carboxylic acids.
4200 compounds
The use of covalently binding inhibitors is steadily growing, with numerous molecules progressing through the stages of clinical trials and even make it to become marketed drugs.
5,816 compounds
Bromodomain Modulators Library is a set of drug-like compounds aimed at modulating PPI of bromodomain-containing proteins with other vital proteins.
20,000 compounds
Chemokine Receptor Targeted Library is a set of small-molecule ligands. Modulation of chemokine receptor is used in the treatment of inflammatory diseases.
9,769 compounds
Set of small-molecule HDAC inhibitors. HDAC regulate gene expression and its inhibitors act against cancers, neurodegenerative and inflammatory diseases.
21,000 compounds
Epitranscriptome Focused Small Molecule Library modulates the activity of proteins involving in aberrant RNA modification.
50,410 compounds
Anti-Aging Library is small molecules targeting cellular pathways and biological targets that are implicated in aging.
29,000 compounds
RNA Isosteric Trinucleotide Mimetics is small molecules targeting RNA expansion repeats. Trinucleotide repeats overexpression causes various disorders.
1,503 compounds
3D Mimetics PPI Library is a set of small-molecule compounds that mimic key recognition elements of protein secondary structure.
9,753 compounds
Indole Derivatives Library is indole-based compounds. These heterocyclic compounds are active molecules with anti-inflammatory effects.
12,563 compounds
Set consists of sp3-enriched β-lactams, generic library of covalent inhibitors, smart library of covalent inhibitors, smart library of covalent fragments.
90,769 compounds
Beyond the Flatland Library sp3-enriched is a set of saturated small-molecules with chemical properties for a faster transition of compounds from discovery to drugs.
4,063 compounds
3D Fragment Library is a set of small-molecule compounds with diverse and well-developed 3D-shapes for HTS and fragment-based drug discovery.
11,269 compounds
Fragments Library is a set of small-molecules with high diversity, reduced structural complexity, drug-likeness. They possess a potential for "fragment evolution” and “fragment linking".
2,109 compounds
ChemDiv's Crystallographic and 19F NMR fragment libraries contain Fluorine Fragments (1480 compounds) and Bromine Fragments (629 compounds). The fragment library consists of small-molecule compounds containing fluorine or bromine atoms. These fragments are well suited for high throughput screening based on fluorine NMR or X-ray crystallography.
799 compounds
Smart library of covalent inhibitors and fragments with a wide range of reactivity warheads.
4,561 compounds
Natural-Product-Based Library is a set of small-molecule compounds. Natural products have proven successful modulators of difficult targets.
Tags
Custom ChemistryNovel Scaffolds and Discovery LibrariesCustom Building Blocks for DNA Encoded LibrariesScale up SynthesisMacrocycle CompoundsIn silico Drug Design (CADD)PROTACADME, DMPKMedicinal ChemistryDNA Encoded Libraries-CDI-CapabilitiesDiscovery BiologyAssay DevelopmentHigh Throughput Screening (HTS)Animal ModelsToxicology and SafetyChemistry, Manufacturing and ControlsPre-Plated SetRepresentative CompoundsNatural-Product3D-PharmacophoreMCE-18RepresentativeSoluble DiversityTargeted DiversitySmartTMAntiviralGPCR3DPhenotypic ScreeningCNS activityTranscription FactorsDrugs LibraryTarget ActivityTherapeutical DiversityCNSIon ChannelsProteases HumanKinases HumanPhosphatases HumanReceptors HumanOpportunistic PathogensCancerCardiovascularMetabolicImmune systemInfectionsMusculoskeletalDigestive systemRespiratory tractOtorhinolaryngologicNervous systemEyeMaleFemaleHemic and lymphaticCongenitalSkinEndocrineAnimalWoundsKinasesProteasesPhosphatasesNuclear receptorsOthersPPI modulatorsReceptor's ligandsEpigeneticMimeticsCyclic compoundsFragmentsPoolChemical classes AgroAllosteric Inhibitors