Masupirdine free base
Chemical Structure Depiction of
Masupirdine free base
Masupirdine free base
Compound characteristics
| Compound ID: | CE01-3235 |
| Compound Name: | Masupirdine free base |
| Molecular Weight: | 478.41 |
| Molecular Formula: | C21 H24 Br N3 O3 S |
| CAS Number: | 701205-60-9 |
| Smiles: | CN1CCN(CC1)Cc1cn(c2ccc(cc12)OC)S(c1ccccc1[Br])(=O)=O |
| InChI Key: | GWCYPEHWIZXYFZ-UHFFFAOYSA-N |
| Short Description: | Masupirdine free base (SUVN-502 free base) is a potent, selective, and orally bioavailable 5-HT6 receptor antagonist with a Ki of 2.04 nM for the human 5-HT6 receptor, demonstrating high selectivity o ver the 5-HT2A receptor and other 100 target sites. It is also brain penetrant and has potential for the treatment of Alzheimer's disease. |
| Pathway: | Neuroscience|||GPCR/G Protein |
| Target: | 5-HT Receptor |
| Alias: | SUVN-502 free base |
| Stock amount: | 997 |