DNA Encoded Libraries-CDI-Capabilities
ChemDiv proposes design and synthesis of heterocyclic scaffolds for DEL:
Vast diversity of heterocyclic scaffolds,
Proprietary and continuously validated reactions and library protocols
High Fsp3 scaffolds
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Flexible and conformationally constrained cores
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Derivatives and mimics of natural compounds
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Poly-functional derivatization
Multiple diversity points, ≥ 3
Defined chirality
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Confirmed relative stereochemistry
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Confirmed absolute stereochemistry
Protein-Protein Interaction modulation as a focus:
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Macrocycles
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Spiro-cycles
- Natural templates