Anti-Inflammatory Library
ChemDiv’s Anti-Inflammatory Library contains 28,000 compounds.
Target space for anti-inflammatory effect includes
1) Chemokines
2) TNF
3) TLR7
4) Kinases (Jak1, Itk, IRAK-4)
5) PDE4
6) P2X7
7) NF-kB
8) Others
Library Statistics:
Number of Scaffolds 654
Unique Heterocycles 544
Diversity Coefficient 0,8416
Number of Screens 10355
MW 175-600; 393 av.
PSA 18-207; 82 av.
Target space for anti-inflammatory effect includes
1) Chemokines
2) TNF
3) TLR7
4) Kinases (Jak1, Itk, IRAK-4)
5) PDE4
6) P2X7
7) NF-kB
8) Others
Library Statistics:
Number of Scaffolds 654
Unique Heterocycles 544
Diversity Coefficient 0,8416
Number of Screens 10355
MW 175-600; 393 av.
PSA 18-207; 82 av.