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Human Kinases Annotated Library

2,500 Compounds

• Kinases are enzymatic proteins that phosphorylate other functional proteins
• Physiologically the kinase enzymatic activity can be modulated by
– Catalytic ATP site binders
– Allosteric binders that cause conformational changes within the catalytic ATP site
• Kinases are well recognized as important therapeutic targets for
– Oncology, e.g. cancer immunotherapy
– Inflammatory diseases, e.g. fibrosis, rheumatoid arthritis
– Cardiovascular system, e.g. cerebral vasospasm, pulmonary arterial hypertension
A unique collection of small molecule compounds with annotated activities for Kinases protein targets
❑ Annotated activities : 236 kinase targets
❑ Express Delivery : 640 compounds
❑ Complete Version : 2585 compounds

Medicinal and Computational Chemistry Dept., ChemDiv, Inc.
12760 High Bluff Dr, San Diego, CA, 92130
Phone: + 1 916 234 0888
Fax: +1 858 794 4931
Email: ChemDiv@chemdiv.com

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